Compile Data Set for Download or QSAR
Found 42 of ic50 data for polymerid = 50003596
TargetHomeodomain-interacting protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50563555(CHEMBL4750420)copy SMILES
Affinity DataIC50: 38nMAssay Description:Inhibition of human recombinant HIPK3 using myelin substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD22MPPubMed
TargetHomeodomain-interacting protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50172243(CHEMBL3103192)copy SMILEScopy InChI
Affinity DataIC50: 40nMAssay Description:Inhibition of Hipk3 (unknown origin) by quantitative PCRMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2C53NRMPubMed
TargetHomeodomain-interacting protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50335638(5-(3-Chlorophenylamino)benzo[c][2,6]naphthyridine-...)copy SMILEScopy InChI
Affinity DataIC50: 45nMAssay Description:Inhibition of recombinant human HIPK3 in presence of ATP at Km concentration by radiometric filter-binding assayMore data for this Ligand-Target Pair
TargetHomeodomain-interacting protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50335638(5-(3-Chlorophenylamino)benzo[c][2,6]naphthyridine-...)copy SMILEScopy InChI
Affinity DataIC50: 45nMAssay Description:Inhibition of human recombinant HIPK3 by radiometric assayMore data for this Ligand-Target Pair
TargetHomeodomain-interacting protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50563541(CHEMBL4743730)copy SMILES
Affinity DataIC50: 65nMAssay Description:Inhibition of human recombinant HIPK3 using myelin substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD22MPPubMed
TargetHomeodomain-interacting protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50563556(CHEMBL4743939)copy SMILES
Affinity DataIC50: 66nMAssay Description:Inhibition of human recombinant HIPK3 using myelin substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD22MPPubMed
TargetHomeodomain-interacting protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM17055((18S)-18-[(dimethylamino)methyl]-17-oxa-4,14,21-tr...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Inhibition of HIPK3 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD22MPPubMed
TargetHomeodomain-interacting protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM16673(4-[4-({[4-chloro-3-(trifluoromethyl)phenyl]carbamo...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Inhibition of HIPK3 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD22MPPubMed
TargetHomeodomain-interacting protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50242737((R,Z)-5-(2,6-dichlorobenzylsulfonyl)-3-((3,5-dimet...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Inhibition of HIPK3 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD22MPPubMed
TargetHomeodomain-interacting protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50399540(FORETINIB | US10464902, Foretinib | US10882853, Co...)copy SMILEScopy InChI
Affinity DataIC50: 100nMAssay Description:Inhibition of HIPK3 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD22MPPubMed
TargetHomeodomain-interacting protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50563538(CHEMBL4797457)copy SMILES
Affinity DataIC50: 125nMAssay Description:Inhibition of human recombinant HIPK3 using myelin substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD22MPPubMed
TargetHomeodomain-interacting protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50563554(CHEMBL4790030)copy SMILES
Affinity DataIC50: 128nMAssay Description:Inhibition of human recombinant HIPK3 using myelin substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD22MPPubMed
TargetHomeodomain-interacting protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50563539(CHEMBL4762964)copy SMILES
Affinity DataIC50: 128nMAssay Description:Inhibition of human recombinant HIPK3 using myelin substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD22MPPubMed
TargetHomeodomain-interacting protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50560704(CHEMBL4754195)copy SMILES
Affinity DataIC50: 159nMAssay Description:Inhibition of human recombinant HIPK3 using myelin substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD22MPPubMed
TargetHomeodomain-interacting protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50560704(CHEMBL4754195)copy SMILES
Affinity DataIC50: 159nMAssay Description:Inhibition of human HIPK3 by radiometric assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GQ72GZPubMed
TargetHomeodomain-interacting protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50563537(CHEMBL4789951)copy SMILES
Affinity DataIC50: 164nMAssay Description:Inhibition of human recombinant HIPK3 using myelin substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD22MPPubMed
TargetHomeodomain-interacting protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)copy SMILEScopy InChI
Affinity DataIC50: 202nMAssay Description:Inhibition of human HIPK3 using MBP as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DJ5KB8PubMed
TargetHomeodomain-interacting protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50563534(CHEMBL4778153)copy SMILES
Affinity DataIC50: 283nMAssay Description:Inhibition of human recombinant HIPK3 using myelin substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD22MPPubMed
TargetHomeodomain-interacting protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50563535(CHEMBL4791451)copy SMILES
Affinity DataIC50: 300nMAssay Description:Inhibition of human recombinant HIPK3 using myelin substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD22MPPubMed
TargetHomeodomain-interacting protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50563540(CHEMBL4740998)copy SMILES
Affinity DataIC50: 441nMAssay Description:Inhibition of human recombinant HIPK3 using myelin substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD22MPPubMed
TargetHomeodomain-interacting protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50563533(CHEMBL4777288)copy SMILES
Affinity DataIC50: 476nMAssay Description:Inhibition of human recombinant HIPK3 using myelin substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetHomeodomain-interacting protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50563536(CHEMBL4741919)copy SMILES
Affinity DataIC50: 692nMAssay Description:Inhibition of human recombinant HIPK3 using myelin substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD22MPPubMed
TargetHomeodomain-interacting protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)copy SMILEScopy InChI
Affinity DataIC50: 710nMAssay Description:Inhibition of human HIPK3 using MBP as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W380MTPubMed
TargetHomeodomain-interacting protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50563551(CHEMBL4777533)copy SMILES
Affinity DataIC50: 720nMAssay Description:Inhibition of human recombinant HIPK3 using myelin substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD22MPPubMed
TargetHomeodomain-interacting protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50563544(CHEMBL4778370)copy SMILES
Affinity DataIC50: 807nMAssay Description:Inhibition of human recombinant HIPK3 using myelin substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD22MPPubMed
TargetHomeodomain-interacting protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50563543(CHEMBL4794825)copy SMILES
Affinity DataIC50: 1.23E+3nMAssay Description:Inhibition of human recombinant HIPK3 using myelin substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD22MPPubMed
TargetHomeodomain-interacting protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50563553(CHEMBL4795812)copy SMILES
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of human recombinant HIPK3 using myelin substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD22MPPubMed
TargetHomeodomain-interacting protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50563552(CHEMBL4747520)copy SMILES
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of human recombinant HIPK3 using myelin substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD22MPPubMed
TargetHomeodomain-interacting protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50563550(CHEMBL4793177)copy SMILES
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of human recombinant HIPK3 using myelin substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD22MPPubMed
TargetHomeodomain-interacting protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50563548(CHEMBL4790254)copy SMILES
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of human recombinant HIPK3 using myelin substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD22MPPubMed
TargetHomeodomain-interacting protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50563547(CHEMBL4747210)copy SMILES
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of human recombinant HIPK3 using myelin substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD22MPPubMed
TargetHomeodomain-interacting protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50563546(CHEMBL4758047)copy SMILES
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of human recombinant HIPK3 using myelin substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD22MPPubMed
TargetHomeodomain-interacting protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50563545(CHEMBL4777540)copy SMILES
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of human recombinant HIPK3 using myelin substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD22MPPubMed
TargetHomeodomain-interacting protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50563542(CHEMBL4789373)copy SMILES
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of human recombinant HIPK3 using myelin substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD22MPPubMed
TargetHomeodomain-interacting protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50563549(CHEMBL4800422)copy SMILES
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of human recombinant HIPK3 using myelin substrate by radiometric scintillation assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD22MPPubMed
TargetHomeodomain-interacting protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50135286(CHEMBL3745885)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human HIPK3 using MBP as substrateMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24Q7WT8PubMed
TargetHomeodomain-interacting protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50001733(CHEMBL3133821)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human HIPK3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TM7CN0PubMed
TargetHomeodomain-interacting protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50519662(CHEMBL4438748)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human recombinant HIPK3 (161 to 562 residues) using myelin basic protein as substrate after 40 mins by [gamma-33ATP] radiometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MC93FGPubMed
TargetHomeodomain-interacting protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM13533(1-[2-(4-methylphenyl)-5-tert-butyl-pyrazol-3-yl]-3...)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of HIPK3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NC61NHPubMed
TargetHomeodomain-interacting protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50359359(CHEMBL1929238)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of HIPK3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NC61NHPubMed
TargetHomeodomain-interacting protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50537742(CHEMBL4634634 | US11179389, Compound 1-14)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant human His-tagged HIPK3 catalytic domain expressed in baculovirus expression system using serine/threonine-9 peptide as subs...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HM5CZGPubMed
TargetHomeodomain-interacting protein kinase 3(Homo sapiens (Human))TBA
LigandPNGBDBM50614163(CHEMBL5288779)copy SMILES
Affinity DataIC50: 9.00E+5nMMore data for this Ligand-Target Pair
Ligand InfoPDB
In DepthDetails